DY268CAS号: 1609564-75-1分子式: C30H32N4O5S分子量: 560.66描述纯度储存/保存方法可溶性/溶解性靶点
产品描述 | |
描述 |
DY268 is a compound based on trisubstituted pyrazolamide without any FXR agonist activity and cytotoxicity and can be used as an effective FXR antagonist (IC50 = 7.5 nM).
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纯度 |
98%
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储存/保存方法 |
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
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基本信息 | |
可溶性/溶解性 |
H2O:Insoluble,DMSO:50 mg/mL (89.18 mM)
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生物活性 | |
靶点 |
FXR:7.5 nM
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