ML 254CAS号： 1428630-86-7分子式： C18H15FN2O2分子量： 310.32描述纯度储存/保存方法可溶性/溶解性靶点
| 产品描述 | |
| 描述 |
ML254 competitively interacts with the MPEP allosteric binding site. ML254 is highly selective for mGlu5 versus other mGlu receptors, has a clean ancillary Ricerca profile, and suitable dystrophia myotonica protein kinase (DMPK) properties for systemic dosing in rodents.
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| 纯度 |
98%
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| 储存/保存方法 |
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
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| 基本信息 | |
| 可溶性/溶解性 |
DMSO:27.5 mg/mL (88.62 mM)
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| 生物活性 | |
| 靶点 |
rat mGluR5:8.03 nM (pEC50), rat mGluR5:9.3 nM (EC50)
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