MK 212盐酸盐CAS号： 64022-27-1分子式： C8H11CIN4.HCl分子量： 235.12描述应用纯度储存/保存方法形态外观熔点沸点折射率IC50Ki 数据可溶性/溶解性MDLPubChem CIDEC号码
| 产品描述 | |
| 描述 |
MK 212 hydrochloride is a SR-2C agonist.
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| 应用 |
A SR-2C agonist
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| 纯度 |
≥99%
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| 储存/保存方法 |
Store at room temperature
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| 形态 |
Solid
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| 基本信息 | |
| 外观 |
Crystalline
|
| 熔点 |
300° C (dec.)
|
| 沸点 |
364.1° C at 760 mmHg (Predicted)
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| 折射率 |
n20D 1.57 (Predicted)
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| IC50 |
SR-2C: EC5050 = 213 nM (human); SR-2B: EC5050 = 295 nM (human)
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| Ki 数据 |
Serotonin 1b (5-HT1b) receptor: Ki= 178 nM (rat); Serotonin 1a (5-HT1a) receptor: Ki= 202 nM (rat); Adrenergic receptor alpha-1: Ki= 913 nM (rat); Serotonin 2 (5-HT2) receptor: Ki= >1 µM (rat); Dopamine D1Ʊᩄ 悐瓒 러Ŕ쬈ශ P Ӥ 러ŔȀ P Ӥ 懀Ȁ
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| 可溶性/溶解性 |
Soluble in water (50 mM), and DMSO (≥20 mg/ml).
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| MDL |
MFCD00673963
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| PubChem CID |
198421
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| EC号码 |
262-883-0
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